Molecule Details
InChIKeyMRWUTTXEVGWLFR-UHFFFAOYSA-N
Compound Name9-[5-(1-methylindazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-4-yl]-2,9-diazaspiro[5.5]undecan-1-one
Canonical SMILESCn1ncc2cc(-c3cnc4[nH]ccc4c3N3CCC4(CCCNC4=O)CC3)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.52
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24863 CCNC Homo sapiens Human PF16899 PF00134 8.5 IC50 ChEMBL;BindingDB
P49336 CDK8 Homo sapiens Human PF00069 8.5 IC50 ChEMBL
Q9BWU1 CDK19 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB