Molecule Details
InChIKeyMRIBBXXALNMJDD-UHFFFAOYSA-N
Compound Name4-[4-[1-(6-methoxypyrimidin-4-yl)-8-[(3-methyl-2-pyridinyl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]phenyl]-N-methylbenzamide
Canonical SMILESCNC(=O)c1ccc(-c2ccc(N3C(=O)N(c4cc(OC)ncn4)C4(CCN(Cc5ncccc5C)CC4)C3=O)cc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96KS0 EGLN2 Homo sapiens Human PF13640 9.5 IC50 ChEMBL;BindingDB
Q9GZT9 EGLN1 Homo sapiens Human PF13640 PF01753 9.3 IC50 ChEMBL;BindingDB
Q9H6Z9 EGLN3 Homo sapiens Human PF13640 7.8 IC50 ChEMBL;BindingDB