Molecule Details
InChIKeyMQTMFZBGEJWSRJ-WDYNHAJCSA-N
Canonical SMILESO=C1CN2CCN(CC2)CC(=O)Nc2ccc(cc2)C[C@@H](NS(=O)(=O)Cc2ccccc2)C(=O)N[C@H](C(=O)O)Cc2ccc(cc2)N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00747 PLG Homo sapiens Human PF00051 PF00024 PF00089 9.2 Ki ChEMBL;BindingDB
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 6.5 Ki ChEMBL;BindingDB