Molecule Details
InChIKeyMQRPDUHCJZKKNO-UHFFFAOYSA-N
Compound Name4-(3,4-dichlorophenyl)-1,1-dimethyl-7-[6-(trifluoromethyl)pyridazin-3-yl]-3,4-dihydro-2H-isoquinoline
Canonical SMILESCC1(C)NCC(c2ccc(Cl)c(Cl)c2)c2ccc(-c3ccc(C(F)(F)F)nn3)cc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.13
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 7.6 IC50 ChEMBL;BindingDB
Q01959 SLC6A3 Homo sapiens Human PF00209 7.5 IC50 ChEMBL;BindingDB
P23975 SLC6A2 Homo sapiens Human PF00209 6.3 IC50 ChEMBL;BindingDB