Molecule Details
InChIKeyMQPHXDFBKUCNOD-BKFWDETESA-N
Canonical SMILESCOc1ccc(NC(=O)c2nc3ccccc3n([C@@H]3C[C@H]4CC[C@@H](C3)N4C3CCCCCCC3)c2=O)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5TC84 OGFRL1 Homo sapiens Human PF04664 6.9 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB