Molecule Details
InChIKeyMPHUHAKFOBHHJK-UHFFFAOYSA-N
Compound Name5-[5-Amino-2-[(2,6-difluorophenyl)methyl]-7-(4-fluorophenyl)-[1,2,4]triazolo[1,5-c]pyrimidin-8-yl]-1-(2-hydroxyethyl)pyridin-2-one
Canonical SMILESNc1nc(-c2ccc(F)cc2)c(-c2ccc(=O)n(CCO)c2)c2nc(Cc3c(F)cccc3F)nn12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.44
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 9.7 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB