Molecule Details
InChIKeyMOYYMSNZEWQWQJ-UHFFFAOYSA-N
Compound Name4-(4-methoxy-2-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)pyridin-2-amine
Canonical SMILESCOc1nc(C)nc2[nH]cc(-c3ccnc(N)c3)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.53
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13627 DYRK1A Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
Q9Y463 DYRK1B Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
Q92630 DYRK2 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB