Molecule Details
InChIKeyMOYQBNCJLIJEOA-UHFFFAOYSA-N
Compound Name6-(2,6-difluorophenyl)-N-(4-piperidin-4-yloxy-3-pyridinyl)pyridine-2-carboxamide
Canonical SMILESO=C(Nc1cnccc1OC1CCNCC1)c1cccc(-c2c(F)cccc2F)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB