Molecule Details
InChIKeyMOQYJMVBPKWDGC-UXHICEINSA-N
Compound Nametrans-(1S,2S)-N-[4-(1-propan-2-ylpyrazol-4-yl)sulfonylphenyl]-2-pyridin-3-ylcyclopropane-1-carboxamide
Canonical SMILESCC(C)n1cc(S(=O)(=O)c2ccc(NC(=O)[C@H]3C[C@@H]3c3cccnc3)cc2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43490 NAMPT Homo sapiens Human PF18127 PF04095 8.3 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.7 IC50 ChEMBL
P11712 CYP2C9 Homo sapiens Human PF00067 6.1 IC50 ChEMBL;BindingDB