Molecule Details
InChIKeyMOFRXFLSGOVYKC-UHFFFAOYSA-N
Compound Name2,2,2-Trifluoro-1-(5-{[(4-methoxyphenyl)methoxy]methyl}thiophen-2-yl)ethan-1-one
Canonical SMILESCOc1ccc(COCc2ccc(C(=O)C(F)(F)F)s2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.39
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P56524 HDAC4 Homo sapiens Human PF12203 PF00850 6.4 pIC50 TTD_MultiTarget
Q02161 RHD Homo sapiens Human PF00909 6.4 pIC50 TTD_MultiTarget
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 6.4 IC50 ChEMBL;BindingDB