Molecule Details
InChIKeyMOAUKNBJAKYOML-KRWDZBQOSA-N
Compound Name3-[4-[(3R)-3-aminopyrrolidin-3-yl]phenyl]-2-(2H-tetrazol-5-yl)-6-(trifluoromethyl)benzenesulfon-amide
Canonical SMILESN[C@@]1(c2ccc(-c3ccc(C(F)(F)F)c(S(N)(=O)=O)c3-c3nn[nH]n3)cc2)CCNC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.46
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 9.3 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 8.1 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.0 IC50 BindingDB