Molecule Details
InChIKeyMNYODQSAKDAGDY-UHFFFAOYSA-N
Compound Name5-chloro-3-methyl-N-(2-methyl-4-piperazin-1-ylquinolin-6-yl)-1-benzothiophene-2-sulfonamide
Canonical SMILESCc1cc(N2CCNCC2)c2cc(NS(=O)(=O)c3sc4ccc(Cl)cc4c3C)ccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.17
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P50406 HTR6 Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB