Molecule Details
InChIKeyMNHWODGSAAWVCT-UHFFFAOYSA-N
Compound Name2,4-Diamino-5-methylpyrido(2,3-d)pyrimidine, 6-((3-methylphenylthio)methyl), 0.7 hydrate
Canonical SMILESCc1cccc(SCc2cnc3nc(N)nc(N)c3c2C)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 6.1 IC50 ChEMBL;BindingDB
O30463 folA Mycobacterium avium Pathogen PF00186 7.8 IC50 ChEMBL
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 7.2 IC50 ChEMBL;BindingDB