Molecule Details
InChIKeyMMGHHQMLYUHLGS-UHFFFAOYSA-N
Compound NameN-[(4-carbamimidoylphenyl)methyl]-2-[5-chloro-2-oxo-3-(pentan-3-ylamino)-6-phenyl-1,2-dihydropyrazin-1-yl]acetamide
Canonical SMILESCCC(CC)Nc1nc(Cl)c(-c2ccccc2)n(CC(=O)NCc2ccc(C(=N)N)cc2)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08709 F7 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 6.4 IC50 ChEMBL;BindingDB
P13726 F3 Homo sapiens Human PF09294 PF01108 6.4 IC50 ChEMBL
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.0 IC50 ChEMBL;BindingDB