Molecule Details
InChIKeyMMFLOBKIGRXPRE-UHFFFAOYSA-N
Compound Name5-fluoro-2-[5-[(sulfamoylamino)methyl]-1,3,4-oxadiazole-2-carbonyl]-N-(2,2,2-trifluoroethyl)-1,3-benzothiazole-6-carboxamide
Canonical SMILESNS(=O)(=O)NCc1nnc(C(=O)c2nc3cc(F)c(C(=O)NCC(F)(F)F)cc3s2)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11150 LIPC Homo sapiens Human PF00151 PF01477 8.4 IC50 ChEMBL;BindingDB
Q9Y5X9 LIPG Homo sapiens Human PF00151 PF01477 7.3 IC50 ChEMBL;BindingDB