Molecule Details
InChIKeyMMCVYWQYORICCQ-UHFFFAOYSA-N
Compound Name8-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-morpholino-1H-1,2,4-triazol-1-yl)phenyl)quinazolin-2-amine
Canonical SMILESCn1cc(-c2cccc3cnc(Nc4ccc(-n5cnc(N6CCOCC6)n5)cc4)nc23)cn1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.39
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P05412 JUN Homo sapiens Human PF00170 PF03957 6.5 IC50 ChEMBL;BindingDB