Molecule Details
InChIKeyMKVQVZUHJKLKRR-UHFFFAOYSA-N
Compound Name5-(furan-2-yl)-6-(pyrimidin-4-yl)-1H-imidazo[4,5-b]pyridin-2(3H)-one
Canonical SMILESO=c1[nH]c2cc(-c3ccncn3)c(-c3ccco3)nc2[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB