Molecule Details
InChIKeyMKVLTWPKSBOTOH-UHFFFAOYSA-N
Compound Name7-cyclopentyl-2-[4-[[7-(hydroxyamino)-7-oxoheptyl]carbamoyl]anilino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide
Canonical SMILESCN(C)C(=O)c1cc2cnc(Nc3ccc(C(=O)NCCCCCCC(=O)NO)cc3)nc2n1C1CCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13547 HDAC1 Homo sapiens Human PF00850 8.8 IC50 ChEMBL;BindingDB
P11802 CDK4 Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
P30281 CCND3 Homo sapiens Human PF02984 PF00134 7.9 IC50 ChEMBL