Molecule Details
InChIKeyMKRNFARKVGJOOC-UHFFFAOYSA-N
Compound Name6-naphthalen-1-ylsulfanyl-5-propan-2-yl-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine
Canonical SMILESCC(C)c1c(Sc2cccc3ccccc23)[nH]c2nc(N)nc(N)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 6.9 IC50 ChEMBL;BindingDB
P0ABQ4 folA Escherichia coli (strain K12) Pathogen PF00186 6.8 IC50 ChEMBL