Molecule Details
InChIKeyMJJJRRMQCUUKEO-IZZDOVSWSA-N
Compound Name(E)-N-(3-((6-(1H-Indol-3-yl)pyrimidin-4-yl)amino)phenyl)-4-(4-(dimethylamino)but-2-enamido)benzamide
Canonical SMILESCN(C)C/C=C/C(=O)Nc1ccc(C(=O)Nc2cccc(Nc3cc(-c4c[nH]c5ccccc45)ncn3)c2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q8TBX8 PIP4K2C Homo sapiens Human PF01504 8.3 Kd ChEMBL;BindingDB
Q9Y2I7 PIKFYVE Homo sapiens Human PF00118 PF00610 PF01363 PF01504 7.4 IC50 ChEMBL;BindingDB
P48426 PIP4K2A Homo sapiens Human PF01504 6.0 IC50 ChEMBL;BindingDB