Molecule Details
InChIKeyMJHMGTYNRCLWJK-UHFFFAOYSA-N
Compound Name5-[2-Chloro-4-(3-methyl-1H-pyrazol-1-yl)benzoyl]-1-methyl-1,4,5,10-tetrahydro pyrazolo[3,4-b][1,5]benzodiazepine
Canonical SMILESCc1ccn(-c2ccc(C(=O)N3Cc4cnn(C)c4Nc4ccccc43)c(Cl)c2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.63
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30559 OXTR Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P37288 AVPR1A Homo sapiens Human PF00001 PF08983 7.6 Ki ChEMBL;BindingDB
P30518 AVPR2 Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB