Molecule Details
InChIKeyMJCKUHBSAUHVJE-UHFFFAOYSA-N
Compound Name1-(6-Morpholin-4-ylpyridin-2-yl)-3-[8-(trifluoromethyl)quinolin-4-yl]urea
Canonical SMILESO=C(Nc1cccc(N2CCOCC2)n1)Nc1ccnc2c(C(F)(F)F)cccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL7.5
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P49840 GSK3A Homo sapiens Human PF00069 8.0 Ki ChEMBL
P49841 GSK3B Homo sapiens Human PF00069 8.0 Ki ChEMBL
P68400 CSNK2A1 Homo sapiens Human PF00069 7.3 Ki ChEMBL
Q8NE63 HIPK4 Homo sapiens Human PF00069 6.7 Ki ChEMBL