Molecule Details
InChIKeyMHWGNSVLNNQWIZ-UHFFFAOYSA-N
Compound Name5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine
Canonical SMILESCCc1nc2[nH]ncc2c2nc(-c3ccccc3)nn12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P0DMS8 ADORA3 Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.6 IC50 ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 6.5 IC50 ChEMBL;BindingDB