Molecule Details
InChIKeyMHSIRMSFRHMBDY-UHFFFAOYSA-N
Compound NameN-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(2-fluoro-3-methoxyphenyl)pyrimidin-4-yl]acetamide
Canonical SMILESCOc1cccc(-c2cc(NC(C)=O)nc(-n3nc(C)cc3C)n2)c1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.09
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 9.2 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB