Molecule Details
InChIKeyMHNMEERHZSPWFL-VSGBNLITSA-N
Compound Name4-[(1R)-1-amino-1-(3-methylimidazol-4-yl)ethyl]-2-[3-[(3R)-3-ethyl-1-methyl-2-oxoazepan-3-yl]phenoxy]benzonitrile
Canonical SMILESCC[C@]1(c2cccc(Oc3cc([C@@](C)(N)c4cncn4C)ccc3C#N)c2)CCCCN(C)C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49356 FNTB Homo sapiens Human PF00432 8.1 IC50 ChEMBL
P49354 FNTA Homo sapiens Human PF01239 7.3 IC50 ChEMBL;BindingDB
P53609 PGGT1B Homo sapiens Human PF00432 7.3 IC50 ChEMBL