Molecule Details
InChIKeyMHNMEERHZSPWFL-NSOVKSMOSA-N
Compound Name2-[3-(3-Ethyl-1-methyl-2-oxo-azepan-3-YL)-phenoxy]-4-[1-amino-1-(1-methyl-1H-imidizol-5-YL)-ethyl]-benzonitrile
Canonical SMILESCC[C@@]1(c2cccc(Oc3cc([C@](C)(N)c4cncn4C)ccc3C#N)c2)CCCCN(C)C1=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.63
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 10.2 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 10.2 IC50 ChEMBL;BindingDB
P53609 PGGT1B Homo sapiens Human PF00432 8.4 IC50 ChEMBL