Molecule Details
InChIKeyMHKGSIVWVNSWNG-UHFFFAOYSA-N
Compound Name2-Methyl-5-(2-{4-[3-pyridin-4-ylbenzyl]piperidin-1-yl}ethoxy)quinoline
Canonical SMILESCc1ccc2c(OCCN3CCC(Cc4cccc(-c5ccncc5)c4)CC3)cccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB