Molecule Details
InChIKeyMHJTWQKANDHIIB-UHFFFAOYSA-N
Compound Name2-(4-fluorophenyl)-6,10-dimethoxy-1H-benzo[h]quinolin-4-one
Canonical SMILESCOc1cc2c(=O)cc(-c3ccc(F)cc3)[nH]c2c2c(OC)cccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16678 CYP1B1 Homo sapiens Human PF00067 8.4 IC50 ChEMBL;BindingDB
P04798 CYP1A1 Homo sapiens Human PF00067 8.0 IC50 ChEMBL;BindingDB
P05177 CYP1A2 Homo sapiens Human PF00067 6.7 IC50 ChEMBL;BindingDB