Molecule Details
InChIKeyMHBGRNASPWNGMV-UHFFFAOYSA-N
Compound Name1-(6-Piperazin-1-yl-2-pyridinyl)-6-(6-prop-1-ynylpyrazin-2-yl)pyrazolo[4,3-c]pyridine
Canonical SMILESCC#Cc1cncc(-c2cc3c(cn2)cnn3-c2cccc(N3CCNCC3)n2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 10.6 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 10.2 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.8 Ki ChEMBL;BindingDB