Target not found.
Molecule Details
InChIKeyMGYNRIYGDOFIPG-UHFFFAOYSA-N
Compound Name5-[[4-(4-Amino-6,7-dimethoxyquinazolin-2-yl)piperazine-1-carbothioyl]amino]-2-(3-hydroxy-6-oxoxanthen-9-yl)benzoic acid
Canonical SMILESCOc1cc2nc(N3CCN(C(=S)Nc4ccc(-c5c6ccc(=O)cc-6oc6cc(O)ccc56)c(C(=O)O)c4)CC3)nc(N)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.91
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 8.0 IC50 ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 7.6 IC50 ChEMBL;BindingDB