Molecule Details
InChIKeyMGXQLLRKRSAUPY-UHFFFAOYSA-N
Compound NameRac-4-((2,3-dichlorophenoxy)(piperidin-4-yl)methyl)pyridine
Canonical SMILESClc1cccc(OC(c2ccncc2)C2CCNCC2)c1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P23975 SLC6A2 Homo sapiens Human PF00209 8.1 IC50 ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 8.1 IC50 ChEMBL;BindingDB
Q01959 SLC6A3 Homo sapiens Human PF00209 7.2 IC50 ChEMBL;BindingDB