Molecule Details
InChIKeyMGLLPZGTTQFMEG-UHFFFAOYSA-N
Compound NameN'-hydroxy-N-[1-(3-methoxypropylamino)isoquinolin-7-yl]octanediamide
Canonical SMILESCOCCCNc1nccc2ccc(NC(=O)CCCCCCC(=O)NO)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O15379 HDAC3 Homo sapiens Human PF00850 7.9 IC50 ChEMBL;BindingDB
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 7.9 IC50 ChEMBL;BindingDB
Q13547 HDAC1 Homo sapiens Human PF00850 7.5 IC50 ChEMBL;BindingDB