Molecule Details
InChIKeyMGJOAQODMQCCGV-UHFFFAOYSA-N
Compound Name3-(4-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-7-methoxybenzofuran-2-yl)-N-(2-(dimethylamino)ethyl)benzamide
Canonical SMILESCOc1cc2c(cc1OC)CN(Cc1ccc(OC)c3oc(-c4cccc(C(=O)NCCN(C)C)c4)cc13)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.98
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18825 ADRA2C Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB