Molecule Details
InChIKeyMGCUTECDFDAQCK-NRFANRHFSA-N
Compound NameC-(3-{2-[(S)-3-(Benzylamino-methyl)-pyrrolidin-1-yl]-ethyl}-1H-indol-5-yl)-N-methyl-methanesulfonamide
Canonical SMILESCNS(=O)(=O)Cc1ccc2[nH]cc(CCN3CC[C@@H](CNCc4ccccc4)C3)c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.4 IC50 ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB