Molecule Details
InChIKeyMGCPJSMHKDVTGW-UHFFFAOYSA-N
Compound Name3-[(4-(4-Fluoro-2-methoxyphenyl)-1,3,5-triazin-2-yl)amino]-benzene-methanesulfonamide
Canonical SMILESCOc1cc(F)ccc1-c1ncnc(Nc2cccc(CS(N)(=O)=O)c2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.96
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O60563 CCNT1 Homo sapiens Human PF00134 PF21797 8.0 IC50 ChEMBL;BindingDB
P50750 CDK9 Homo sapiens Human PF00069 8.0 IC50 ChEMBL