Molecule Details
InChIKeyMFWHDFGMXHATNR-UHFFFAOYSA-N
Compound Name2,9-Dimethyl-5-[(1-piperidin-4-ylpyrazol-4-yl)amino]-2,4,6,9-tetrazatetracyclo[9.8.0.03,8.013,18]nonadeca-1(19),3,5,7,11,13,15,17-octaen-10-one
Canonical SMILESCN1C(=O)c2cc3ccccc3cc2N(C)c2nc(Nc3cnn(C4CCNCC4)c3)ncc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60285 NUAK1 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
Q9UQB9 AURKC Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB