Molecule Details
InChIKeyMERYTOPZZMIEFD-UCQJWODQSA-N
Compound Namebenzyl N-[(2S)-1-[(2S)-2-[[2,2-dimethyl-1-[(2S,6R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]butyl]carbamoyl]pyrrolidin-1-yl]-1-oxo-3,3-diphenylpropan-2-yl]carbamate
Canonical SMILESCCC(C)(C)C(NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)OCc1ccccc1)C(c1ccccc1)c1ccccc1)B1O[C@@H]2CC3CC(C3(C)C)[C@]2(C)O1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 10.5 Ki ChEMBL;BindingDB
P00747 PLG Homo sapiens Human PF00051 PF00024 PF00089 7.5 Ki ChEMBL;BindingDB
P08311 CTSG Homo sapiens Human PF00089 7.4 Ki ChEMBL;BindingDB