Molecule Details
InChIKeyMEHDKDKCBBBTSM-YEWWUXTCSA-N
Canonical SMILESC[C@@](NC(=O)c1ccsc1)(c1cn(CC#N)nn1)[C@H]1CC[C@H](C)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P25774 CTSS Homo sapiens Human PF08246 PF00112 9.0 IC50 ChEMBL;BindingDB
P07711 CTSL Homo sapiens Human PF08246 PF00112 6.0 IC50 ChEMBL;BindingDB