Molecule Details
InChIKeyMDMMWSVMDMOFFW-UHFFFAOYSA-N
Compound Name3-ethyl-N-(4-methoxyphenyl)-3-methyl-2,5-dioxo-1,4-dihydro-1,4-benzodiazepine-7-sulfonamide
Canonical SMILESCCC1(C)NC(=O)c2cc(S(=O)(=O)Nc3ccc(OC)cc3)ccc2NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q10469 MGAT2 Homo sapiens Human PF05060 8.4 IC50 ChEMBL;BindingDB
P26572 MGAT1 Homo sapiens Human PF03071 7.5 IC50 ChEMBL;BindingDB