Molecule Details
InChIKeyMDCMULVKRBERMG-UHFFFAOYSA-N
Compound NameN-(4-(2-(4-(1H-1,2,3-Triazol-1-yl)phenylamino)pyrimidin-4-yl)-phenyl)methanesulfonamide
Canonical SMILESCS(=O)(=O)Nc1ccc(-c2ccnc(Nc3ccc(-n4ccnn4)cc3)n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.1
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB