Molecule Details
InChIKeyMBGVUMXBUGIIBQ-LEWJYISDSA-N
Compound Name1-((3R,4R)-1-(Cyclooctylmethyl)-3-(hydroxymethyl)-4-piperidinyl)-3-ethyl-1,3-dihydro-2H-benzimidazol-2-one
Canonical SMILESCCn1c(=O)n([C@@H]2CCN(CC3CCCCCCC3)C[C@H]2CO)c2ccccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.32
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41146 OPRL1 Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 6.7 Ki BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 6.6 Ki BindingDB