Molecule Details
InChIKeyMAXWOEDRRCSRHI-OALUTQOASA-N
Compound Name(6S,7S)-6-[4-(3-ethylphenyl)-3,6-dihydro-2H-pyridine-1-carbonyl]-N-hydroxy-5-azaspiro[2.5]octane-7-carboxamide
Canonical SMILESCCc1cccc(C2=CCN(C(=O)[C@H]3NCC4(CC4)C[C@@H]3C(=O)NO)CC2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.15
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 7.7 pIC50 TTD_MultiTarget
O14672 ADAM10 Homo sapiens Human PF21299 PF00200 PF13574 7.0 IC50 ChEMBL;BindingDB
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 6.7 IC50 ChEMBL;BindingDB