Molecule Details
InChIKeyLZYWVOKHWFMDJU-UHFFFAOYSA-N
Compound Name2-amino-5-(3-ethyl-1H-pyrrolo[2,3-b]pyridin-5-yl)-N,N-dimethylbenzamide
Canonical SMILESCCc1c[nH]c2ncc(-c3ccc(N)c(C(=O)N(C)C)c3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q92918 MAP4K1 Homo sapiens Human PF00780 PF00069 8.7 Ki ChEMBL;BindingDB
P00519 ABL1 Homo sapiens Human PF08919 PF07714 PF00017 PF00018 7.7 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.3 IC50 ChEMBL;BindingDB