Molecule Details
InChIKeyLZPFBEBTZBKKFB-UHFFFAOYSA-N
Compound Name19-(3-Methoxyphenyl)-1,14,16,22-tetrazatricyclo[13.5.2.018,21]docosa-15,17,19,21-tetraen-6-ol
Canonical SMILESCOc1cccc(-c2cn3c4nc(ncc24)NCCCCCCCC(O)CCCC3)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.39
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q12866 MERTK Homo sapiens Human PF00041 PF00047 PF13927 PF07714 6.8 IC50 ChEMBL;BindingDB
P36888 FLT3 Homo sapiens Human PF00047 PF07714 6.3 IC50 ChEMBL;BindingDB
P30530 AXL Homo sapiens Human PF00041 PF13927 PF07714 6.0 IC50 ChEMBL;BindingDB