Molecule Details
InChIKeyLZKXNZXRQFFQAH-UHFFFAOYSA-N
Compound Name2-amino-N-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-phenylacetamide
Canonical SMILESNC(C(=O)Nc1cc2cc[nH]c(=O)c2cc1Cl)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.98
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O75116 ROCK2 Homo sapiens Human PF25346 PF00069 PF08912 7.4 IC50 ChEMBL;BindingDB
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 7.2 IC50 ChEMBL;BindingDB
Q16513 PKN2 Homo sapiens Human PF02185 PF00069 PF00433 6.3 IC50 ChEMBL;BindingDB