Molecule Details
InChIKeyLYMPHEWUZFSXGM-UHFFFAOYSA-N
Compound Name9-cyclopentyl-8-N-(2-fluorophenyl)-2-N-methylpurine-2,8-diamine
Canonical SMILESCNc1ncc2nc(Nc3ccccc3F)n(C3CCCC3)c2n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.3
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P45984 MAPK9 Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB