Molecule Details
InChIKeyLYIMJKFUHYOWBM-UHFFFAOYSA-N
Compound Name6-Fluoro-4-[[2-hydroxy-3-[4-(1,6-naphthyridin-5-yl)piperazin-1-yl]propyl]amino]chromen-2-one
Canonical SMILESO=c1cc(NCC(O)CN2CCN(c3nccc4ncccc34)CC2)c2cc(F)ccc2o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P0AES4 gyrA Escherichia coli (strain K12) Pathogen PF03989 PF00521 6.8 IC50 ChEMBL;BindingDB
P0AFI2 parC Escherichia coli (strain K12) Pathogen PF03989 PF00521 6.7 IC50 ChEMBL;BindingDB