Molecule Details
InChIKeyLXUURPGAYDBQPD-UHFFFAOYSA-N
Compound Name6-N-methyl-6-N-(3,4,5-trimethoxyphenyl)pyrido[2,3-d]pyrimidine-2,4,6-triamine
Canonical SMILESCOc1cc(N(C)c2cnc3nc(N)nc(N)c3c2)cc(OC)c1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 8.3 IC50 ChEMBL;BindingDB
P16184 Pneumocystis carinii Pathogen PF00186 8.6 IC50 ChEMBL