Molecule Details
InChIKeyLXFPTSIBSQOGTO-AREMUKBSSA-N
Compound Name(2r)-2-[(1-Aminoisoquinolin-6-Yl)amino]-4,11-Diazatricyclo[14.2.2.1~6,10~]henicosa-1(18),6(21),7,9,16,19-Hexaene-3,12-Dione
Canonical SMILESNc1nccc2cc(N[C@H]3C(=O)NCc4cccc(c4)NC(=O)CCCc4ccc3cc4)ccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P06870 KLK1 Homo sapiens Human PF00089 7.7 Ki ChEMBL;BindingDB
P08709 F7 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 6.4 Ki ChEMBL;BindingDB
P13726 F3 Homo sapiens Human PF09294 PF01108 6.4 Ki ChEMBL