Molecule Details
InChIKeyLWULHXVBLMWCHO-UHFFFAOYSA-N
Compound NameSR142948A
Canonical SMILESCOc1cccc(OC)c1-c1cc(C(=O)NC2(C(=O)O)C3CC4CC(C3)CC2C4)nn1-c1ccc(C(=O)N(C)CCCN(C)C)cc1C(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.44
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30990 NTS Homo sapiens Human PF07421 9.6 Ki BindingDB
P30989 NTSR1 Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB
O95665 NTSR2 Homo sapiens Human PF00001 7.1 Ki ChEMBL